Chemotherapy medicine bottle melting under intense heat, symbolizing cancer treatment issues.

Doxorubicin and Thermal Ablation: Do Chemo Drugs Survive the Heat?

"A new study investigates if the chemotherapy drug doxorubicin remains effective after thermal ablation, a common cancer treatment."


For individuals battling liver cancer, combined transarterial chemoembolization (TACE) and percutaneous thermal ablation has emerged as a powerful treatment option. TACE delivers chemotherapy directly to the tumor site, while thermal ablation uses heat to destroy cancerous cells. The combined approach aims to maximize the destruction of tumors while minimizing side effects. But a crucial question remains: does the chemotherapeutic drug, specifically doxorubicin (DOX), survive the extreme heat of thermal ablation?

The effectiveness of TACE followed by thermal ablation hinges on whether the chemotherapy drug can withstand the heat. If the drug degrades during the ablation process, the potential benefits of the combined approach may be limited. Understanding the thermal effects on locally delivered chemotherapeutic drugs is therefore essential for optimizing cancer treatment strategies.

To investigate this critical question, a new ex vivo study was undertaken to test the hypothesis that doxorubicin chemotherapy can survive thermal ablative heating. This research provides valuable insights into the stability of doxorubicin under thermal stress, potentially impacting how combined cancer treatments are planned and executed.

Doxorubicin's Fate Under Fire: What the Study Revealed

Chemotherapy medicine bottle melting under intense heat, symbolizing cancer treatment issues.

The study, published in Diagnostic and Interventional Radiology, directly challenged the initial assumption that doxorubicin survives thermal ablation unscathed. Researchers Joseph D. Morrison, Collin K. Schlager, Amanda E. Lee, Richard B. van Breemen, and Ron C. Gaba designed an experiment to mimic the conditions of combined TACE and thermal ablation outside of a living organism.

The researchers submerged fresh porcine (pig) psoas major muscle tissue in a doxorubicin solution to simulate TACE, allowing the tissue to become saturated with the drug. The tissue was then subjected to microwave ablation (MWA) at a controlled temperature, mimicking the thermal ablation process. Finally, the concentration of doxorubicin in the tissue was carefully measured using a sophisticated technique called ultra-high performance liquid chromatography tandem mass spectrometry (UHPLC-MS/MS).

  • Unexpected Results: Contrary to the initial hypothesis, the study found that tissue doxorubicin concentration progressively decreased with increasing ablation time.
  • Quantifiable Degradation: Longer exposure to microwave ablation led to a significant reduction in the amount of doxorubicin present in the tissue.
  • Statistical Significance: Differences in tissue doxorubicin levels between unablated tissue and MWA groups were statistically significant (P < 0.001).
These findings suggest that the heat from thermal ablation may break down doxorubicin, reducing its concentration and potentially its effectiveness. The implication is that TACE followed by ablation might result in lower intratumoral doxorubicin levels than if TACE were used alone.

Implications for Cancer Treatment: What Does This Mean for Patients?

The study's findings raise important questions about the optimal sequencing and delivery of combined TACE and thermal ablation. If thermal ablation reduces doxorubicin concentration, clinicians may need to adjust treatment protocols to ensure sufficient drug exposure to cancer cells. This could involve:

<ul> <li><b>Adjusting drug dosages:</b> Clinicians might consider increasing the initial dose of doxorubicin during TACE to compensate for potential degradation during ablation.</li> <li><b>Optimizing ablation techniques:</b> Exploring alternative ablation methods or adjusting ablation parameters (e.g., duration, power) to minimize heat-induced drug degradation could be beneficial.</li> <li><b>Exploring alternative drugs:</b> Researching alternative chemotherapeutic agents that are more resistant to thermal degradation may offer a more effective combined treatment strategy.</li> </ul>

While this ex vivo study provides valuable insights, further research is needed to confirm these findings in living organisms. In vivo studies can account for factors such as blood flow and drug metabolism, which could influence the degradation of doxorubicin during thermal ablation. Further research may also be warranted in an in vivo animal model system to assess whether the effects are retained in living systems, and whether intraparenchymal DOX concentrations remain at cytotoxic levels following thermal ablation after delivery at standard therapeutic dosing. Despite these limitations, this research highlights the importance of understanding the interplay between chemotherapy and thermal ablation to optimize cancer treatment outcomes.

About this Article -

This article was crafted using a human-AI hybrid and collaborative approach. AI assisted our team with initial drafting, research insights, identifying key questions, and image generation. Our human editors guided topic selection, defined the angle, structured the content, ensured factual accuracy and relevance, refined the tone, and conducted thorough editing to deliver helpful, high-quality information.See our About page for more information.

This article is based on research published under:

DOI-LINK: 10.5152/dir.2018.17382, Alternate LINK

Title: Does Doxorubicin Survive Thermal Ablation? Results Of An Ex Vivo Bench Top Study

Subject: Cardiology and Cardiovascular Medicine

Journal: Diagnostic and Interventional Radiology

Publisher: AVES Publishing Co.

Authors: Joseph D. Morrison, Collin K. Schlager, Amanda E. Lee, Richard B. Van Breemen, Ron C. Gaba

Published: 2018-01-09

Everything You Need To Know

1

What is the focus of the study?

The study investigated the effectiveness of the chemotherapy drug, doxorubicin, after thermal ablation. Thermal ablation is a cancer treatment that uses heat to destroy tumors, often used in conjunction with Transarterial Chemoembolization (TACE). The combined approach aims to maximize tumor destruction while minimizing side effects for liver cancer patients.

2

What are Transarterial Chemoembolization (TACE) and thermal ablation, and how are they related?

Transarterial Chemoembolization (TACE) delivers chemotherapy drugs, like doxorubicin, directly to the tumor site. Thermal ablation uses heat to destroy cancerous cells. The study was designed to understand if doxorubicin, delivered via TACE, remains effective when followed by thermal ablation. If doxorubicin degrades during the ablation process, the benefits of the combined approach may be limited.

3

What were the main findings of the research regarding doxorubicin and thermal ablation?

The research found that doxorubicin concentration decreased with increasing ablation time. The longer the tissue was exposed to microwave ablation, the less doxorubicin was present. These findings suggest that the heat from thermal ablation breaks down doxorubicin, potentially reducing its effectiveness in treating cancer.

4

What does the study's results mean for cancer treatment?

The implications of this study suggest that the sequencing and delivery of Transarterial Chemoembolization (TACE) and thermal ablation might need adjustment. If thermal ablation reduces doxorubicin levels, clinicians may need to alter treatment protocols to ensure adequate drug exposure to cancer cells. This could involve adjusting the timing of the treatments or modifying drug dosages.

5

Why are the study's findings important?

The study's findings are significant because they challenge the initial assumptions about the combined use of Transarterial Chemoembolization (TACE) and thermal ablation. The research demonstrates that doxorubicin, a key chemotherapy drug, may not survive the heat generated during thermal ablation. This impacts how clinicians plan and execute cancer treatments, particularly for liver cancer. The study used microwave ablation (MWA) to simulate the thermal ablation process and ultra-high performance liquid chromatography tandem mass spectrometry (UHPLC-MS/MS) to measure the doxorubicin levels.

Newsletter Subscribe

Subscribe to get the latest articles and insights directly in your inbox.